Description
NM-2201
Product information
IUPAC-name Naphthalen-1-yl 1-(5-fluoropentyl)-1H-indole-3-carboxylate
Synonyms CBL-2201
Formal name naphthalen-
Cas number 837122-21-7
Formula C24H22FNO2
Molar Mass 375.443 g·mol−1
Formulation Powder
Solubility
- Dichloromethane: 20 mg/ml
- DMF: 20 mg/ml
- DMSO: 20 mg/ml
- Ethanol: 5 mg/m
Shipping & Storage Information
NM-2201 which is also known as CBL-2201 is an analytical reference standard compound that is categorized as a synthetic cannabinoid. Specifically, it is an indole-based synthetic cannabinoid, with similar characteristics to 5F-PB-22 and NNE1. The N-fluoropentyl indole core is linked to the N-phthalene ring through an ester bond. This structure is similar to that of 5F-PB-22. Like the 5F-PB-22, it contains a naphthalene ring and a quinoline ring. The chemical structure is similar to AM-2201, but it differs from the latter in that its linkage has changed from carbonyl to ester. NM-2201 is an analog of the AM-2201 a potent synthetic cannabinoid with Ki values of 1.0 and 2.6 nM for CB1 and CB2 receptors respectively. The linkage between naphthalene and its indole core became linked to the ester in AM-2201.
NM-2201 is an indole-based synthetic cannabinoid that is a presumably full agonist. It binds the CB1 and CB2 receptors with low nanomolar affinity. It is a highly potent cannabinoid, with Ki values of 1.0 and 2.6 nM for central cannabinoid receptors.
NM-2201 is a full agonist that has a binding affinity of 0.80 nM at CB1 and 0.35 nM at CB2.
The toxicological and physiological properties of this compound has not been analyzed. Due to the lack of sufficient safety and pharmacology data for SCs, human pharmacokinetic studies are typically not conducted. This issue is most apparent in the lack of published data for compounds such as AM-2201. Usage of this Chemical should be for research and forensic purposes only.
NM-2201 is classified as a Schedule I substance due to its high potential for abuse and its lack of accepted medical uses. The substance is not approved for human use in the United States and is not intended to be consumed or tested on humans. However, it may be useful for forensic purposes. It was originally discovered in 1989 at the Northeastern University, where it is now manufactured. It is one of the most potent synthetic cannabinoids in common use.
WARNING This product is not for human or veterinary use.
This product is only available to persons of 21 years old and above.
Hazard statement(s)
| H302 | Harmful if swallowed |
| H315 | Causes skin irritation |
| H319 | Causes serious eye irritation |
| H332 | Harmful if inhaled |
| H335 | May cause respiratory irritation |
| H336 | May cause drowsiness or dizziness |
| Precautionary statement(s) | |
| P264 | Wash hands thoroughly after handling |
| P280 | Wear protective gloves/protective clothing/eye protection/face protection |
| P305 + P351 + P338 | IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing. |
| P337 + P313 | If eye irritation persists: Get medical advice/attention |
| P261 | Avoid breathing dust/ fume/ gas/ mist/ vapors/ spray |
| P271 | Use only outdoors or in a well-ventilated area |
| P304 + P340 | IF INHALED: Remove victim to fresh air and keep at rest in a position comfortable for breathing |
| P312 | Call a POISON CENTER or doctor/physician if you feel unwell |
| P403 + P233 | Store in a well-ventilated place. Keep container tightly closed |
| P405 | Store locked up |
| P501 | Dispose of contents/container to a licensed disposal company |
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